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Qi Xu, Ning Wu, Xiangqian Li, Chuanlong Guo, Chao Li, Bo Jiang, Huaizhi Wang, Dayong Shi*. Inhibition of PTP1B blocks pancreatic cancer progression by targeting the PKM2/AMPK/mTOC1 pathway.Cell Death & Disease.2019. (IF=5.959)accepted
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Guo, Chuanlong; Wang, Lijun; Li, Xiuxue; Wang, Shuaiyu; Yu, Xuemin; xu, kuo; Zhao, Yue; Luo, Jiao; Li, Xiangqian; Jiang, Bo; Shi, Dayong*. Discovery of novel bromophenol - thiosemicarbazone hybrids as potent selectve inhibitors of poly(ADP-ribose) polymerase-1 (PARP1) for use in cancer.Journal of Medicinal Chemistry.2019, 62, 6, 3051-3067. (IF=6.253)
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Xiangqian Li, Qi Xu, Chao Li, Jiao Luo, Lijun Wang, Bo Jiang, Dayong Shi*. Uncharged Bromophenol improves insulin sensitivity in BKS db mice through selective inhibition of PTP1B.European Journal of Medicinal Chemistry 2019,166 , 178-185. (IF=4.816)
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Wang, Lijun; Guo, Chuanlong; Li, Xiuxue; Luo, Jiao; Li, Xiangqian; Jiang, Bo; Shi, Dayong*. Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment.European Journal of Medicinal Chemistry2019,177, 1:153-170 (IF=4.816)
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Jiao Luo, Qi Xu, Bo Jiang, Renshuai Zhang, Xiaoling Jia, Xiangqian Li, Lijun Wang, Chuanlong Guo, Ning Wu, Dayong Shi*.Selectivity, cell permeability and oral availability studies of novel bromophenol derivative HPN as PTP1B inhibitor. Br. J. Pharmacol.2018, 75: 140–153.(IF=6.810)
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Lina Ma, Xiaolin Shi, Xiaowei Li, Dayong Shi*. Iron-catalyzed alkynylation of tertiary aliphatic amines with 1-iodoalkkynes to synthesize propargylamines.Organic Chemistry Frontiers.2018,00:1-5. (IF=5.455)
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Wu, Ning; Zhang , Chunyun; Wang, Changhui; Yao, Weicheng; Song, Lairong; Lin, Xiukun; Shi, Dayong*. Zinc-Doped Copper Oxide Nanocomposites reverse Temozolomide resistance in Glioblastoma by inhibits AKT and ERK1/2.Nanomedicine. 2018,13(11): 1303–1318. (IF=5.005)
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Li Ning, Wang Lijun, Jiang Bo, Li Xiangqian, Guo Shuju, Shi, D.-Y.*, Recent progress of the development of dipeptidyl peptidase-4 inhibitors for the treatment of type 2 diabetes mellitus.European Journal of Medicinal Chemistry. 2018, 151, 145-157. (IF=4.816)
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Renshuai Zhang, Rilei Yu, Qi Xu, Xiangqian Li, Jiao Luo, Bo Jiang, Lijun Wang, ShujuGuo, NingWua, Dayong Shi*. Discovery and evaluation of the hybrid of bromophenol and saccharide as potent and selective protein tyrosine phosphatase 1B inhibitors.European Journal of Medicinal Chemistry. 2017; 134:24-33. (IF=4.816)
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Xiangqian Li, Qi Xu, Jiao Luo, Lijun Wang, Bo Jiang, Renshuai Zhang, Dayong Shi*.Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B. European Journal of Medicinal Chemistry. 2017; 136:348-359. (IF=4.816)